PI3-K alpha Inhibitor 2 (Echelon Product Code: B-0304 1MG)
| Description: | 3-(4-Morpholinothieno[3, 2-d]pyrimidin-2-yl)phenol is a selective inhibitor for the "-isoform of PI 3-Kinase (IC(50): PI 3-K" = 2 nM, PI 3-K" = 16 nM, PI3-K" = 660 nM, PI3KC2" = 220 nM)). It showed 1000-fold selectivity vs. protein kinases such as PKA, KDR, PKCa, and E/CDK2 (IC(50) = 91, 3.4, 466, 288 µM). It inhibited proliferation of A375 melanoma cells at 580 nM. Also known as PI3-K Inhibitor 2, PIK2. » References; 1) M. Hayakawa, et al. "Synthesis and biological evaluation of 4-morpholino-2-phenyl quinazolines and related derivatives as novel PI3 kinase p110a inhibitors" Bioorg. Med. Chem. 2006, 14, 6847-6858. |
| Order #: | ECH-B-0304-1MG |
| Unit Size: | 1 mg |
| Supplier: | Echelon Biosciences |
| Restrictions: | Available in all European countries, except France & Italy. |
| Shipping: | Room Temperature |
| Storage: | 4-8 °C |
| Subcategory: | Biochemical Reagents |
| More information: | Go to webpage |
87.00 € *
*All prices are net in Euro and do not include applicable taxes, shipping & handling, or other charges (e.g., customs duties).
Delivery time approx. 8 - 10 working days
- Phone: +49 (0)89 3799666-6
- Fax: +49 (0)89 3799666-99
- E-mail: order@biozol.de
- Online Shop: www.mobitec.com
- Phone: +49 (0)89 3799666-6
- E-mail: info@biozol.de
How To Order
Orders can be placed by phone, fax, e-mail, or via our online shop:
MoBiTec is now part of BIOZOL
All orders and requests placed via the online shop on www.mobitec.com are processed by BIOZOL Diagnostica Vertrieb GmbH.
You will receive an order confirmation by fax or e-mail. More information regarding the ordering process can be found here.
Technical Service - Product Information
Viewed